5-(2-Pyrimidinyl)-imidazo[1,2-a]pyridines are antibacterial agents targeting the ATPase domains of DNA gyrase and topoisomerase IV

5-(2-Pyrimidinyl)-imidazo[1,2-a]pyridines are antibacterial agents targeting the ATPase domains of DNA gyrase and topoisomerase IV DNA gyrase (GyrB)/topoisomerase IV (ParE) inhibitors: Synthesis and antibacterial activity New N -phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity Fragment-to-Hit-to-Lead Discovery of a Novel Pyridylurea Scaffold of ATP Competitive Dual Targeting Type II Topoisomerase Inhibiting Antibacterial Agents Novel Dual-Targeting Benzimidazole Urea Inhibitors of DNA Gyrase and Topoisomerase IV Possessing Potent Antibacterial Activity: Intelligent Design and Evolution through the Judicious Use of Structure-Guided Design and Stucture−Activity Relationships Discovery of Pyrazolopyridones as a Novel Class of Gyrase B Inhibitors Using Structure Guided Design Design, synthesis, and structure–activity relationship studies of ATP analogues as DNA gyrase inhibitors Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors Dual Targeting of GyrB and ParE by a Novel Aminobenzimidazole Class of Antibacterial Compounds An optimised series of substituted N-phenylpyrrolamides as DNA gyrase B inhibitors