New class of potent ligands for the human peripheral cannabinoid receptor

Bioorganic & Medicinal Chemistry Letters
1996.0

Abstract

A new class of potent ligand for the human peripheral cannabinoid (hCB2) receptor is described. Two indole analogs 13 and 17 exhibited nanomolar potencies (Ki) with good selectivity for the hCB2 receptor over the human central cannabinoid (hCB0 receptor. Copyright © 1996 Elsevier Science Ltd

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