Structure–activity relationships of α-amino acid ligands for the α2δ subunit of voltage-gated calcium channels

Structure–activity relationships of α-amino acid ligands for the α2δ subunit of voltage-gated calcium channels N-Acridin-9-yl-butane-1,4-diamine derivatives: high-affinity ligands of the α2δ subunit of voltage gated calcium channels Part 1: N-Alkylated glycines as potent α2δ ligands Structure−Activity Relationships of Pregabalin and Analogues That Target the α₂-δ Protein Investigation into the preferred conformation of gabapentin for interaction with its binding site on the α2δ subunit of a calcium channel Synthesis and in vivo evaluation of 3-substituted gababutins Ca²⁺Channel α₂-δ Ligands for the Treatment of Neuropathic Pain Novel Cyclopropyl β-Amino Acid Analogues of Pregabalin and Gabapentin That Target the α₂-δ Protein Carboxylate bioisosteres of gabapentin Carboxylate bioisosteres of pregabalin