Investigation into the preferred conformation of gabapentin for interaction with its binding site on the α2δ subunit of a calcium channel

Investigation into the preferred conformation of gabapentin for interaction with its binding site on the α2δ subunit of a calcium channel Synthesis and biological evaluation of conformationally restricted gabapentin analogues Structure–activity relationships of α-amino acid ligands for the α2δ subunit of voltage-gated calcium channels Synthesis and in vivo evaluation of 3-substituted gababutins N-Acridin-9-yl-butane-1,4-diamine derivatives: high-affinity ligands of the α2δ subunit of voltage gated calcium channels Structure−Activity Relationships of Pregabalin and Analogues That Target the α₂-δ Protein Synthesis and in vivo evaluation of 3,4-disubstituted gababutins Carboxylate bioisosteres of gabapentin Carboxylate bioisosteres of pregabalin Novel Cyclopropyl β-Amino Acid Analogues of Pregabalin and Gabapentin That Target the α₂-δ Protein